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. 2023 Dec 14;66(24):16704–16727. doi: 10.1021/acs.jmedchem.3c01406

Table 6. PK Data for Oral Administration in Mice (30 mg/kg)a.

  plasma concentration ng/mL
compound 30 min 60 min 120 min 180 min 300 min
9b 112   13    
43 164 59   42 21
45 99 92   57 47
60 34   19    
63·HCl 1595 608 111 90 60
a

N = 3 per time point.

b

10 mg/kg p.o.