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. 2023 Dec 6;10(1):e23289. doi: 10.1016/j.heliyon.2023.e23289

Table 2.

Kinetic parameters of DPP-IV in the absence/presence of inhibitors.

Kinetic parameter Inhibitor concentration (μg/mL) No inhibitor CBD CBG CBN THC
KM (mM) 0.52
2.5 0.43 0.28 0.85 0.55
5 0.58 0.33 0.63 0.59
10 0.74 0.55 0.68 0.57
20 1.3 0.56 0.5 0.56
Vmax (mM/min) 1.2
2.5 0.61 0.68 1.01 1.1
5 0.59 0.65 0.93 1.8
10 0.55 0.70 0.86 1.0
20 0.51 0.60 0.74 0.97