Table 2.
Kinetic parameters of DPP-IV in the absence/presence of inhibitors.
| Kinetic parameter | Inhibitor concentration (μg/mL) | No inhibitor | CBD | CBG | CBN | THC |
|---|---|---|---|---|---|---|
| KM (mM) | 0.52 | |||||
| 2.5 | 0.43 | 0.28 | 0.85 | 0.55 | ||
| 5 | 0.58 | 0.33 | 0.63 | 0.59 | ||
| 10 | 0.74 | 0.55 | 0.68 | 0.57 | ||
| 20 | 1.3 | 0.56 | 0.5 | 0.56 | ||
| Vmax (mM/min) | 1.2 | |||||
| 2.5 | 0.61 | 0.68 | 1.01 | 1.1 | ||
| 5 | 0.59 | 0.65 | 0.93 | 1.8 | ||
| 10 | 0.55 | 0.70 | 0.86 | 1.0 | ||
| 20 | 0.51 | 0.60 | 0.74 | 0.97 | ||