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. 2023 Dec 29;67(1):81–109. doi: 10.1021/acs.jmedchem.3c00925

Table 10. Antimycobacterial Activities of Compounds T6030, T6053, 67b, 67c, 69c, and 69e against M.tb. H37Ra Overproducing DprE1/2 Expressed as MIC.

  BTZ-043 (ng/mL) T6030 (μM) T6053 (μM) 67b (μM) 67c (μM) 69c (μM) 69e (μM)
pVV2 1 0.3 0.18 0.125 0.5–1.5 3 0.25–0.5
pVV2-dprE1/2 >30 0.09–0.3 0.18 1.5 1.5 1–3 3