Anticancer activity, determined by MTT assays after 72 h treatment. IC50 values (μM) are given as mean ± SD.
| Drugs | HCT116 | CT26 | Panc-1 |
|---|---|---|---|
| IC50 (μM) ± SD | |||
| Gemcitabine | 0.008 ± 0.002 | 0.040 ± 0.004 | >100 |
| Cisplatin | 5.5 ± 1.0 | 3.4 ± 0.5 | 10.7 ± 1.6 |
| CisPt(OAc)2 | 68.7 ± 10.3 | 8.4 ± 0.1 | 90.9 ± 12.8 |
| CisPt-GemCarb-OAc | 0.020 ± 0.002 | 0.15 ± 0.01 | 29.7 ± 5.7 |
| CisPt-GemSucc-OAc | 0.052 ± 0.002 | 0.14 ± 0.03 | 15.7 ± 4.0 |