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. 2023 Dec 6;11(2):534–548. doi: 10.1039/d3qi02032k

Anticancer activity, determined by MTT assays after 72 h treatment. IC50 values (μM) are given as mean ± SD.

Drugs HCT116 CT26 Panc-1
IC50 (μM) ± SD
Gemcitabine 0.008 ± 0.002 0.040 ± 0.004 >100
Cisplatin 5.5 ± 1.0 3.4 ± 0.5 10.7 ± 1.6
CisPt(OAc)2 68.7 ± 10.3 8.4 ± 0.1 90.9 ± 12.8
CisPt-GemCarb-OAc 0.020 ± 0.002 0.15 ± 0.01 29.7 ± 5.7
CisPt-GemSucc-OAc 0.052 ± 0.002 0.14 ± 0.03 15.7 ± 4.0