Figure 5.
Oligomeric sdAb:cd40 variants display strong CD40 agonism. (a) Domain architecture of oligomeric sdAb:CD40 variants. DANA refer to the D256A-N297A mutation preventing/reducing FcγR binding of IgG1. (b) Western blot analysis of reduced sdAb:cd40 variants. Position of MW (kDa) markers are indicated. Asterixes refer to not fully reduced protein species. (c) U2OS cells were stimulated overnight with the different VHH:CD40 variants and finally IL8 production was determined by ELISA. (D,E) the indicated constructs were purified by affinity chromatography and analyzed by SDS-PAGE (D) and gel filtration (E). Dotted arrows indicate flag peptide remained from the affinity purification.