Skip to main content
. 2024 Jan 20;15:645. doi: 10.1038/s41467-024-44874-3

Table 1.

SAR Exploration of compounds 1-6

Compound Structure % Inhibition at 10 μM (SD) IC50 (nM)
1 graphic file with name 41467_2024_44874_Taba_HTML.gif 2 ND
2 graphic file with name 41467_2024_44874_Tabb_HTML.gif 88 ± 2.60 232
3 graphic file with name 41467_2024_44874_Tabc_HTML.gif -1 ND
4 graphic file with name 41467_2024_44874_Tabd_HTML.gif 2 ND
5 graphic file with name 41467_2024_44874_Tabe_HTML.gif 8 ND
6 graphic file with name 41467_2024_44874_Tabf_HTML.gif 95 ± 0.31 119

SD Standard Deviation, ND Not determined.