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. 2023 Nov 27;15(1):355–365. doi: 10.1039/d3md00473b

ADCs with an average DAR of 4.

ADC Linker DAR DAR4 peak HIC RT/min Agg/%
Ab 0 3.37 1.6
ADC1 Ala–Ala 3.8 4.90 1.0
ADC2 Ala–Arg 3.6 4.52 1.1
ADC3 Ala–Gln 3.7 4.83 1.8
ADC4 Ala–Glu 3.3 4.65 1.3
ADC5 Ala–Gly 3.7 4.77 2.1
ADC6 Ala–His 3.5 4.90 1.7
ADC7 Ala–Lys 2.4 4.18 1.9
ADC8 Ala–Ser 4.2 4.82 1.4
ADC9 Gly–Ala 3.8 4.80 1.7
ADC10 Gly–Gln 3.7 4.71 1.3
ADC11 Gly–Glu 3.2 4.57 1.9
ADC12 Gly–Gly 3.6 4.74 1.9
ADC13 Gly–Ser 3.7 4.69 1.3
ADC14 Phe–Lys 3.7 4.68 3.1
ADC15 Ser–Ala 3.8 4.87 1.8
ADC16 Ser–Asn 3.5 4.72 1.5
ADC17 Ser–Gln 3.6 4.79 1.1
ADC18 Ser–Glu 3.5 4.63 1.7
ADC19 Ser–Gly 3.7 4.77 1.8
ADC20 Val–Ala 3.8 5.10 1.3
ADC21 Val–Arg 3.4 4.73 1.7
ADC22 Val–Cit 3.6 4.98 1.2
ADC23 Val–Asn 3.5 4.90 1.1
ADC24 Val–Gln 4.1 5.02 1.3
ADC25 Val–Glu 3.4 4.79 2.0
ADC26 Val–Gly 3.6 4.99 1.3
ADC27 Val–Ser 3.7 4.98 1.5