Comparison of ADC properties by switching P1 and P2 position in the linker.
| ADC | Dipeptide | HIC Ret time/min | Agg/% |
|---|---|---|---|
| ADC44 | Ser–Ala | 6.48 | 4.90 |
| ADC34 | Ala–Ser | 6.42 | 5.00 |
| ADC38 | Gly–Ala | 6.29 | 7.70 |
| ADC32 | Ala–Gly | 6.49 | 7.90 |
| ADC42 | Gly–Ser | 6.14 | 6.20 |
| ADC48 | Ser–Gly | 6.33 | 6.10 |
| ADC36 | Ala–Val | 6.92 | 13.6 |
| ADC49 | Val–Ala | 6.74 | 12.9 |