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. 2023 Dec 25;17(1):32. doi: 10.3390/ph17010032
HRMS High-resolution mass spectrometry;
HPLC High-performance liquid chromatography;
LDA Lithium diisopropylamide;
NMR Nuclear magnetic resonance;
PG Protecting group;
TFA Trifluoroacetic acid.
ER α Estrogen receptor α
AI Aromatase inhibitor
SERM Selective estrogen receptor modulator
SI Selectivity index
GAPDH Glyceraldehyde-3-phosphate dehydrogenase
GREB1 Gene regulated in breast cancer 1 protein
AR Androgen receptor
CDK4 Cyclin-dependent kinase 4
PARP Poly (ADP-ribose) polymerase 1
Bcl-2 B-cell CLL/lymphoma 2
HT 4-hydroxytamoxifen
MDR Multidrug-resistant