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. Author manuscript; available in PMC: 2024 Sep 7.
Published in final edited form as: Bioorg Med Chem. 2023 Jun 29;92:117400. doi: 10.1016/j.bmc.2023.117400

Table 1.

Oxetane-Containing Indole-based Analogues

graphic file with name nihms-1928982-t0009.jpg
Compound R1 R2 R3 R4 R5 Yield
5a H H H H H 23%
5b H Cl H CH3 H 31%
5c H Br H H H 14%
5d OCH3 H H CH3 H 5%
5e H Cl H OCH3 H 17%
5f H Br H CH3 H 34%
5g H H H H OCH3 30%
5h H H OCH3 H H 13%
5i H H H OCH3 H 10%
5j H H H CH3 H 27%
5k H Cl H H H 11%
5l OCH3 H H H H 22%
5m H OCH3 H OCH3 OH 12%
5n Br H H H H 14%