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. 2012 Jul 12;130(3):187–197. doi: 10.1590/S1516-31802012000300009

Table 3. Common medications causing gynecomastia41 .

Type of agent Medications
Antiandrogens Bicalutamide, cyproterone, flutamide, finasteride, spironolactone
Antibiotics Isoniazid, ketoconazole, metronidazole
Antihypertensives Amlodipine, captopril, enalapril, nifedipine, reserpine, verapamil
Chemotherapeutic agents Cyclophosphamide, methotrexate
Diuretic Spironolactone
Gastrointestinal agents Cimetidine, omeprazole, metoclopramide, ranitidine
Hormones Androgens, anabolic steroids, estrogens, growth hormone
Psychiatric agents Diazepam, haloperidol, phenothiazine, tricyclic antidepressants
Others Amiodarone, antiretrovirals, digitalis, domperidone, statins, theophylline