TABLE 1.
Anti-HIV activity against HIV-1 LAI in PBM cellsa
| NRTI | Anti-HIVLAI in PBM (μM)
|
||
|---|---|---|---|
| EC50 | EC90 | IC50 | |
| d4G | 0.34 ± 0.27 | 3.4 ± 1.2 | 54.2 |
| Cyclo-d4G | 1.1 ± 0.06 | 17.0 ± 3.9 | 84.5 |
Values represent the means ± SD of at least three independent experiments done in triplicate.