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. 2024 Jan 31;16(2):210. doi: 10.3390/pharmaceutics16020210

Table 1.

Selected Pharmakon-1600 drugs (106) for in vitro evaluation against O. gutturosa adult male parasites. Bioactivity was categorised by MicroSource Discovery Systems, Inc. (Gaylordsville, CT, USA).

Bioactivity Drug
Antibacterial Carbadox; Cefaclor; Cefamandole nafate; Cefoperazone; Cefoxitin sodium; Cefsulodin sodium; Ceftibuten; Cefuroxime sodium; Chlorhexidine dihydrochloride; Chloroxylenol; Demeclocycline hydrochloride; Doxycycline hydrochloride; Furazolidone; Gramicidin; Lasalocid sodium; Merbromin; Methacycline hydrochloride; Methenamine; Minocycline hydrochloride; Nitrofurantoin; Nitroxoline; Ofloxacin; Oxytetracycline; Rifampcin; Rifaximin; Sulfaquinoxaline sodium; Teicoplanin
Anticancer Azaserine; Bleomycin; Daunorubicin; Doxorubicin; Epirubicin hydrochloride; Isotretinon; Lomustine; Mitoxantrone hydrochloride; Tretinoin
Antihypertensive/
vasodilator
Dipyridamole; Guanethidine; Losartan; Nicardipine hydrochloride; Nicotinyl alcohol tartrate; Nifedipine
Anti-infective Benzethonium chloride; Broxyquinoline; Dequalinium chloride; Methylbenzethonium chloride; Nitrofurazone; Oxyquinoline hemisulfate; Phenylethyl alcohol; Resorcinol monoacetate
Anti-inflammatory/
antihistamine
Dexamethasone acetate; Doxylamine succinate; Meloxicam sodium; Prednisolone tebutate; Sulfasalazine
Antiparasitic Amitraz; Atovaquone; Candicidin; Clorsulon; Diethylcarbamazine citrate; Flubendazole; Hexetidine; Homidium bromide; Iodoquinol; Levamisole hydrochloride; Moxidectin; Primaquine phosphate; Pyrantel pamoate;
Antiviral Oseltamivir phosphate; Valganciclovir hydrochloride
Neurological Acepromazine maleate; Almotriptan; Ampyzine sulfate; Apomorphine hydrochloride; Armodafinil; Bupropion; Chlorpromazine; Danazol; Desipramine hydrochloride; Dopamine hydrochloride; Isradipine (also antihypertensive/vasodilator); Methsuximide; Methylphenidate hydrochloride; Olanzapine; Oxidopamine hydrochloride; Penfluridol; Rivastigmine tartrate; Selegiline hydrochloride; Zaleplon
Various Alendronate sodium; Anisindione; Ascorbyl palmitate; Bromhexine hydrochloride; Butacaine; β-Carotene; Clopidogrel sulfate; Dienestrol; Dioxybenzone; Docusate sodium; Fluorescein; Mangafodipir trisodium; Methylergonovine maleate; Propoxycaine hydrochloride; Riboflavin; Sennoside A; Tetrahydrozoline hydrochloride