| AUC | area under the curve |
| CCK1R | cholecystokinin type 1 receptor |
| CXCR4 | C-X-C chemokine receptor type 4 |
| DAB | diaminobutyric acid |
| DOTA | 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid |
| DOTAGA | 1,4,7,10-tetraazacyclododececane-1-(glutaric acid)-4,7,10-triacetic acid |
| EB | Evans Blue |
| EMA | European Medicines Agency |
| FAP | fibroblast activation protein |
| FAPI | fibroblast activation protein inhibitor |
| FDA | Food and Drug Administration |
| GFK | glycine phenylalanine-lysine |
| GLP-1R | glucagon-like peptide-1 receptor |
| GY | glycine-tyrosine |
| HBED-CC | N,N′-bis-[2-hydroxy-5-(carboxyethyl)benzyl]ethylenediamine-N,N′-diacetic acid |
| HE | histidine-glutamic acid |
| Her2/neu | human epidermal growth factor receptor 2 |
| HYNIC | hydrazinonicotinic acid |
| kDa | kilodalton |
| mAb | monoclonal antibody |
| MAG3 | mercaptoacetylglycylglycylglycin |
| MC1R | melanocortin-1 receptor |
| mCRPC | metastatic castration resistant prostate cancer |
| α-MSH | melanocyte stimulating hormone |
| MVK | methionine-valine-leucine |
| NEP | neutral endopeptidase |
| NODAGA | 1,4,7-triazacyclononane-1-(glutaric acid)-4,7-diacetic acid |
| NOTA | 1,4,7-triazacyclononane-1,4,7-triacetic acid |
| NOTA-p-SCN | S-2-(4-isothiocyanatobenzyl)-1,4,7-triazacyclononane-1,4,7-triacetic acid |
| PEG | polyethylene glycol |
| PET | positron emission tomography |
| PGA | polyglutamic acid |
| p.i. | post injection |
| PSMA | prostate specific membrane antigen |
| RGD | arginine-glycine-aspartic acid |
| sdAb | single-domain antibody-fragment |
| SPECT/CT | single photon emission computed tomography/computed tomography |
| TE2A | 1,4,8,11-tetraazabicyclo[6.6.2]hexadecane-4,11-diacetic acid |
| TRT | targeted radionuclide therapy |
| uPAR | urokinase-type plasminogen receptor |