Table 2.
cAMP Functional Assay Data at hA2AAR and hA3AR Expressed in CHO Cellsa
compound no. | % activation, A2A cAMP assay | % activation, A3 cAMP assay |
---|---|---|
5a | 0.3 ± 0.3 | 16 ± 4 |
5d | 0.8 ± 0.3 | 4 ± 4 |
5g | 0.05 ± 0.1 | 11 ± 5 |
At a concentration of 10 μM, unless noted.