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. Author manuscript; available in PMC: 2024 Sep 14.
Published in final edited form as: J Med Chem. 2023 Aug 21;66(17):12249–12265. doi: 10.1021/acs.jmedchem.3c00806

Table 2.

cAMP Functional Assay Data at hA2AAR and hA3AR Expressed in CHO Cellsa

compound no. % activation, A2A cAMP assay % activation, A3 cAMP assay
5a   0.3 ± 0.3 16 ± 4
5d   0.8 ± 0.3   4 ± 4
5g 0.05 ± 0.1 11 ± 5
a

At a concentration of 10 μM, unless noted.