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. 2023 Dec 30;30(3):218–225. doi: 10.18553/jmcp.2023.23277

TABLE 2.

Therapeutic Alternatives for the 10 Selected Medicare Drugs by FDA-Approved Indication

Drug FDA-approved indication Therapeutic alternative
Eliquis (apixaban) Treatment and prevention of VTEs Dabigatran
Xarelto (rivaroxaban) Warfarin
Nonvalvular atrial fibrillation
Treatment and prevention of stroke
Xarelto (rivaroxaban) Treatment and prevention of VTEs Pradaxa (dabigatran)
Eliquis (apixaban)
Warfarin
Nonvalvular atrial fibrillation
Treatment and prevention of stroke
Reducing the risk of CV events in CAD/PAD
Jardiance (empagliflozin) Reduce the risk of CV death and hospitalizations for patients with HF Invokana (canagliflozin)
Farxiga (dapagliflozin)
Steglatro (ertugliflozin)
Reduce the risk of CV death in patients with T2D and established CVD
Adjunct therapy to diet and exercise to improve glycemic control in patients with T2D
Farxiga (dapagliflozin) Reduce the risk of CV death and hospitalizations for patients with HFrRF Invokana (canagliflozin)
Jardiance (empagliflozin)
Steglatro (ertugliflozin)
Reduce the risk of CV death in patients with T2D and established CVD or multiple cardiovascular risk factors
Adjunct therapy to diet and exercise to improve glycemic control in patients with T2D
Reduce the risk of sustained eGFR decline, ESRD, CV death and hospitalization for HF in adults with CKD at risk of progression
Januvia (sitagliptin) Adjunct to diet and exercise to improve glycemic control in patients with T2D Onglyza (saxagliptin)
Tradjenta (linagliptin)
Nesina (alogliptin)
Farxiga (dapagliflozin)
Invokana (canagliflozin)
Jardiance (empagliflozin)
Steglatro (ertugliflozin)
Bydureon (exenatide)
Adlyxin (lixisenatide)
Trulicity (dulaglutide)
Victoza (liraglutide)
Ozempic (semaglutide)
Fiasp & Novolog (insulin aspart) Glycemic control for diabetes mellitus Humalog (insulin lispro)
Admelog (insulin lispro)
Entresto (sacubitril/valsartan) Reduce the risk of CV death and hospitalization for HF in adults with CHF Captopril
Enalapril
Lisinopril
Ramipril
Candesartan
Losartan
Valsartan
Treatment of symptomatic HF with systemic left ventricular dysfunction
Enbrel (etanercept) Rheumatoid arthritis Adalimumab
Cimzia (certolizumab)
Infliximab
Simponi (golimumab)
Juvenile idiopathic arthritis
Ankylosing spondylitis
Plaque psoriasis
Psoriatic arthritis
Stelara (ustekinumab) Moderate to severe plaque psoriasis Skyrizi (risankizumab)
Active psoriatic arthritis
Moderate to severe Crohn’s disease
Moderate to severe ulcerative colitis
Imbruvica (ibrutinib) Chronic lymphocytic leukemia/small lymphocytic lymphoma Calquence (acalabrutinib)
Brukinsa (zanubrutinib)
Waldenstrom macroglobulinemia
Chronic graft-vs-host disease

ACE = angiotensin-converting enzyme; ARB = angiotensin receptor blocker; CAD = coronary artery disease; CHF = chronic heart failure; CKD = chronic kidney disease; CV = cardiovascular; CVD = cardiovascular disease; FDA = US Food and Drug Administration; HF = heart failure; HFrRF = heart failure with reduced ejection fraction; VTE = venous thromboembolism; PAD = peripheral artery disease; T2D = type 2 diabetes.