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. 2023 Sep 27;14(2):157–176. doi: 10.1016/j.jpha.2023.09.001

Table 2.

Protective effects of herbal medicine extracts on cardiomyocytes.

Extracts Animal/Cells Models Dose/Concentration Effects Related molecular targets
Refs.
Up-regulation Down-regulation
HJT C57BL/6 J mice; H9c2 cells LAD-induced MI/RI 28 μL/10 g Attenuating I/R-induced infarct size; Alleviating cardiac cell apoptosis; Limiting over-expression of autophagy mTOR AMPK [152]
DMF SD rats LAD-induced MI/RI 60 mg/kg/d Ameliorating heart disease AMPK, Sirt1, PGC-1α [153]
PGS SD rats LAD-induced MI 50, 100 mg/kg Reducing necrotic myocardium; Ameliorating cardiac function Sirt1, ERK1/2, p38MAPK, Bcl-2 Bax, TNF-α, NF-κB [154]
PNs C57BL/6J mice LAD-induced HF 10, 100 μg/mL Improving survival ratio of MI mice; Preserving cardiac function; Elevating the autophagy of cardiomyocytes AMPK, CaMKⅡ ULK1 [155]
HHA C57BL/6J mice P407-induced hyperlipidemic 200 mg/kg/day Improving cardiac remodeling; Attenuating oxidative stress; Promoting mitochondrial biogenesis AMPK, PGC-1α [156]
Gg H9c2 cells DOX-induced cardiotoxicity 40 μg/mL Reducing oxidative stress; Improving cardiac morphology Sirt1, PPARα [157]
AOF SD rats d-galactose-induced aging mice 50, 100, 150 mg/kg Improving heart function; Reducing apoptosis Bcl-2, PI3K, AMPK, Sirt1, PGC-1α Bax [158]
PF Zucker lean rats Zucker diabetic fatty rats 500 mg/kg Reducing cardiac TG content and plasma level PPARα, AMPKα2 [159]

SD: Sprague Dawley; HJT: Hongjingtian injection; DMF: dracocephalum moldavica total flavonoids; PGS: saponins extract from panax japonicus; PNs: panax noto ginseng saponins; HHA: Houttuynia cordata herbal extract; Gg: glycyrrhiza glabra; AOF: alpinate oxyphyllae fructus; PF: pomegranate flower; LAD: ligation of the left anterior descending coronary artery; MI/RI: myocardial ischemia-reperfusion injury; mTOR: mammalian target of rapamycin; AMPK: adenosine monophosphate activated protein kinase; Sirt1: silent information regulator 1; PGC-1α: peroxisome proliferator-activated receptor γ coactivator 1α; MI: myocardial ischemia; ERK1/2: extracellular signal-regulated kinase; p38 MAPK: protein 38 mitogen-activated protein kinase; Bcl-2: B-cell lymphoma-2; Bax: Bcl2-associated x; TNF-α: tumor necrosis factor α; NF-κB: nuclear factor-kappa-B; HF: heart failure; CaMK Ⅱ: calmodulin dependent protein kinase Ⅱ; ULK1: unc-51-like kinase 1; HF: heart failure.