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. 2024 Jan 11;9(2):102195. doi: 10.1016/j.esmoop.2023.102195

Table 4.

Emetogenic potential of single oral antineoplastic agentsa

High/moderate Abemaciclib Lenvatinib
Adagrasib Lomustine
Avapritinib Midostaurin
Bosutinib Mobocertinib
Cabozantinib Niraparib
Ceritinib Olaparib
Crizotinib Procarbazine
Cyclophosphamide Ribociclib
Enasidenib Rucaparib
Fedratinib Selinexorb
Hexamethylmelamine (altretamine) Temozolomide
Imatinib Vinorelbine
Low/minimal Acalabrutinib Methotrexate
Afatinib Neratinib
Alectinib Nilotinib
Alpelisib Nintedanib
Apalutamide Olutasidenib
Asciminib Osimertinib
Axitinib Palbociclib
Bexarotene Panobinostat
Brigatinib Pazopanib
Capecitabine Pemigatinib
Capmatinib Pexidartinib
Chlorambucil Pomalidomide
Cobimetinib Ponatinib
Dabrafenib Pralsetinib
Dacomitinib Regorafenib
Darolutamide Relugolix
Dasatinib Ripretinib
Duvelisib Ruxolitinib
Encorafenib Selpercatinib
Entrectinib Sonidegib
Erdafitinib Sorafenib
Erlotinib Sotorasib
Estramustine Sunitinib
Etoposide Talazoparib
Everolimus Tazemetostat
Fludarabine Tegafur–uracil
Futibatinib Tepotinib
Gefitinib Thalidomide
Gilteritinib Tioguanin (6-thioguanine)
Glasdegib Tivozanib
Hydroxyurea Topotecan
Ibrutinib Trametinib
Idelalisib Trifluridine–tipiracil
Infigratinib Tucatinib
Ivosidenib Umbralisib
Ixazomib Vandetanib
Lapatinib Vemurafenib
Larotrectinib Venetoclax
Lenalidomide Vismodegib
Lorlatinib Vorinostat
Melphalan (L-phenylalanine mustard) Zanubrutinib
a

Classified emetic potential of oral agents based on a full course of therapy and not a single dose within the first cycle.

b

Emetic potential appears to be at the high end of the moderate category.