Table 2. EC50 Values and Hill Coefficients (nH) of ACh in the Presence of the Indicated Concentrations of BPCs at Human α7 and (α1)2β1εδ nAChRs.
| compound | α7 |
(α1)2β1εδ |
||||
|---|---|---|---|---|---|---|
| EC50 | 95% CI μMa | nH | EC50 | 95% CI μMa | nH | |
| ACh | 36.5 | 33.5–40.0 | 1.90 | 15.4 | 13.1–18.8 | 1.22 |
| +3 μM MB327 | 43.8 | 33.6–58.2 | 1.66 | |||
| +10 μM MB327 | 13.0 | 8.1–26.1 | 1.10 | |||
| +3 μM PTM0002 | 51.6 | 42.5–63.2 | 1.57 | |||
| +10 μM PTM0007 | 35.8 | 29.2–45.7 | 1.93 | |||
| +3 μM PTM0015 | 49.2 | 31.7–82.2 | 1.53 | |||
| +0.3 μM PTM0022 | 58.8 | 44.0–81.4 | 1.46 | |||
| +1 μM PTM0022 | 10.3 | 7.3–17.2 | 1.06 | |||