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. 2024 Mar 22;12:RP91973. doi: 10.7554/eLife.91973

Table 2. Calculated Kd values of dihydrotetrabenazine (DTBZ) for various single-point mutants.

Mutant Kd (nM)
WT 15±3
N34A ND
N34D ND
N34Q ND
N34T ND
E127A 15±6
F135A ND
R189A ND
V232L ND
E312Q ND
W318A ND
W318F 24±16
W318H ND
W318R ND
F429A 7.7±0.6
Y433A ND