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. 2023 Mar 9;22(6):1129–1143. doi: 10.2174/1570159X21666221229160300

Table 2.

Study characteristics.

Study (Sample Size) Study Design and Setting Percentage of Male Participants Mean Age (SD) of the Participants Number (%) of Cases with a Psychotic Disorder Number (%) of Cases with Other Psychiatric Disorders Abstinence before the Start of the Study Intervention Group(s) Other Interventions Treatment Duration Assessment Time Points Drinking Measures Drinking Outcomes Other Outcomes Completion Rate Results
Self-Report Bio-markers
Disulfiram
Mueser et al., 2003 [19](N = 33) RCROutpatients 64% 37 years (± 7.1) N = 25 (76%)(S: n = 15; SAD: n = 8;UP: n = 1; SPD: n = 1) N = 8 (24%)(BD: n = 5;MDD: n = 3) Not reported Disulfiram 125-500 mg/day AP + OPTNFS < 1 month (n = 4);1-3 months (n = 7); 3-6 months (n = 3); 6-12 months (n = 3); 1-2 years (n = 8); 2-3 years (n = 3): > 3 years (n = 8) 1-, 2-, and 3-years following initiation of disulfiram treatment AUS None AUS, remission from AUD DUS, number of days spent in hospital (per year), number of weeks worked (per year), side effects. 100%(52 weeks) Reduced AUS scores were observed at 1-, 2-, and 3-years follow-up compared to baseline.Remission from AUD was seen in 21 patients (64%) for at least one year during the follow-up period, in 10 patients (30%) for two years, and in 3 patients (10%) for the full three years of follow-up.Reduced DUS scores were observed at 1-, 2-, and 3-years follow-up compared to baseline.A reduction in the number of days spent in the hospital was observed at the 3-year follow-up compared to baseline.Mild to moderate side effects were reported by 7 patients. Alcohol-disulfiram reactions were experienced by 7 patients.
Disulfiram vs. Naltrexone
Petrakis et al., 2005, 2006 [42, 53](N = 254) DB/OL RCT (DB naltrexone/OL disulfiram)Outpatients 97% 47 years (± 8.2) N = 18 (7%)(S/SAD: n = 18) MDD: n = 178 (70%)PTSD: n = 109 (43%)GAD: n = 57 (20%)CUD: n = 50 (22%)BD: n = 49 (19%) min. 3 days; max. 29 days Naltrexone50 mg/day (n = 59) vs.Disulfiram 250 mg/day (n = 66) vs.Naltrexone 50 mg/day+ disulfiram 250 mg/day (n = 65) vs.Placebo (n = 64) AP + OPTNFS 12 weeks Week 12 TLFB GGTSGOTSGPT CDA, DA, DDW, HDD, TA, GGT, SGOT, SGPT OCDS, BSI, side effects (HCSL) 89% Overall, patients treated with either disulfiram or naltrexone had more CDA and fewer DDW post-treatment compared to the placebo group. Disulfiram-treated patients had reduced levels of GGT at post-treatment compared to naltrexone-treated patients. Patients with PD (S, SAD, BD) had fewer CDA and more HDD than those without PD. Also, patients treated with either disulfiram or naltrexone had more DA and fewer HDD compared with a placebo.Overall, disulfiram-treated patients had lower OCDS and BSI scores at post-treatment compared to naltrexone-treated participants.Patients treated with either disulfiram or naltrexone had lower OCDS and BSI scores post-treatment compared to the placebo group.Overall, there was no advantage of combining disulfiram and naltrexone with respect to any of the outcomes. This was also the case among patients with PD.Mild to severe side effects. Symptoms potentially related to side effects were reported by 96.9% of the participants. Patients with PD were more likely to report mild to moderate side effects compared to those without PD.Fourteen adverse events were recorded, 3 in the combined disulfiram and naltrexone group, 6 in the disulfiram group, 1 in the naltrexone group, and 4 in the placebo group. 43% (n = 6) of the adverse events were reported by patients with PD.
Vasile et al., 2013 [43]*(N = 20) OL RCTSetting not reported 45% 40 years (SD not reported)/ N = 20 (100%)(S: n = 20) None Not reported Naltrexone 50 mg/day (n = 8) vs.Disulfiram 250 mg/day (n = 12) AP 24 weeks Week 24 None None None CGI-S, GAF, IDTS-A, PANSS, side effects Max. 75% Both the disulfiram and naltrexone groups exhibited improvements from baseline to post-treatment on all outcomes, with no differences observed between the two groups.Mild to moderate side effects were observed in both the disulfiram (6 patients) and naltrexone (4 patients) groups.
Naltrexone
Maxwell and Shinder-mann 2000 [51](N = 72) RCROutpatients 71% Not reported N = 24 (33%)S: n = 17(23.3%)SAD: n = 7(5.5%) MDD: n = 37(50.7%)BD: n = 11(15.1%)GID: n = 4(4.1%) Not required Naltrexone unknown dose OPTNFS2 8 weeks week 8 Not reported None Reduced drinking Side effects 82% Reduced drinking was observed at post-treatment compared to baseline. Completers reduced their drinking by at least 75%, and only 17% of the patients relapsed after 8 weeks.Mild side effects.
Batki et al., 2007 [49](N = 19) Single-arm, OL trialOutpatients 79% 43 years (±12) N = 19 (100%)(S: n = 11; SAD: n = 7; UP: n = 1) None Not required Naltrexone 350 mg/ week AP + OPTNFS 8 weeks week 4week 8 TLFB CDTGGT DDW, DWDDD, DDI% CDT% GGT ASIVAS (craving and VAS QoH), PANSS, side effects 74% A reduction in DW, DDD, and DDI, as well as in scores on the ASI, VAS, and PANSS, was observed at post-treatment compared to baseline.No associations were found between self-reported drinking outcomes and alcohol biomarkers.Mild to moderate side effects.
Batki et al., 2010 [48]*(N = 25) Single-arm, OL trialOutpatients 52% 44 years (SD not reported) N = 17 (68%)(S :n = 6; SAD: n = 11) N = 8(BD: n = 8) Not reported Extended-release naltrexone 380 mg/ q4wk AP + PI (motivational counselling- weekly sessions) 12 weeks week 12 TLFB (outcome not reported) None DW, DD, HDD, DDD Side effects 84% Significant improvements were observed from baseline to post-treatment with respect to all outcomes.Mild to moderate side effects. One serious adverse event was recorded.
Vasiliu et al., 2020 [52]*(N = 12) RCRInpatients 33% 29 years (SD not reported) N = 12 (100%)(SAD-bipolar type: n = 2; SAD-depressive type: n = 10) None min. 10 days Naltrexone 50mg/day AP Not reported At discharge from hospital 4 weeks after hospital discharge AUDIT None AUDIT score CGI-S, CDSS, GAF, PANSS, side effects Not reported AUDIT and PANSS scores improved from baseline to (1) the time of discharge from the hospital and (2) four weeks after hospital discharge. CGI-S and GAF scores improved from baseline to time of discharge from hospital. CDSS scores improved significantly from baseline to four weeks after hospital discharge.Mild to moderate side effects.
Petrakis et al., 2004 [44](N = 31) DB RCTOutpatients 100% 46 years (± 5.7) N = 31 (100%)(S: n = 18; SAD: n = 13) None Not required Naltrexone 50 mg/day (n = 16) vs.Placebo (n = 15) AP + PI (cognitive behavioral relapse prevention strategies – weekly sessions) 12 weeks week 12 TLFB (used to validate UTS but outcome is not reported) UTS DD, HDD, TDSP TCQ, PANSS, side effects (HSCL) 81% A reduction in DD and HDD at post-treatment was observed in the naltrexone group compared to the placebo group. There was no drug-by-time interaction effect with respect to either DD or HDD. A reduction in TCQ scores at post-treatment was observed in the naltrexone group compared to the placebo group.Mild side effects. A total of 4 adverse events were recorded, 3 in the naltrexone group and 1 in the placebo group.
Batki et al., 2009 [45]* (N = 90) DB RCTOutpatients 71% 42.5 years (SD not reported) N = 90 (100%)(S: n = 45; SAD: n = 45) None Not reported Naltrexone 350 mg/week (n = 45) vs.Placebo (n = 45) PI (motivational counselling- weekly sessions) 12 weeks week 12 TLBF (outcome not reported) None DW, DD, HDD VAS (craving and QoH) Not reported At post-intervention, a reduction in HDD was observed in the naltrexone group compared to the placebo group.Side effects were not examined.
Naltrexone vs. Acamprosate
Bratu and Sopterean 2014 [46]* (N = 36) OL RCTSetting not reported 67% Mean age not reportedAge range: 18-65 years. N = 36 (100%)(S: n = 36) None min. 7 days Naltrexone 50 mg/day (n = 12) vs.Acamprosate 999 mg/day (n = 12) vs.Counselling (n = 12) AP 24 weeks Week 24 Not reported TL DA, HDD, change in TL GAF, IDTS-A, PANSS, side effects Not reported At post-treatment, an increase in DA and a reduction in HDD were observed in both medication groups compared to the counselling group. An increase in DA was observed in the acamprosate group compared to the naltrexone group, but the naltrexone group had fewer HDD than the acamprosate group. Both medication groups also exhibited improved TL scores compared to the counselling group.Both naltrexone and acamprosate treatment were well tolerated, with no severe adverse effects.
Acamposate
Ralevski et al., 2011 [47] (N = 23) DB RCTOutpatients 83% 51 years (±7.3) N = 23 (100%)(S: n = 9, SAD: n = 10; UP: n = 4) None min. 5 days; max. 21 days Acamprosate 1998 mg/day (n = 12)Placebo (n = 11) AP + PI (skills training in relapse prevention) 12 weeks Week 12 TLFB None ASP, CDA, DD, DDD, HDD OCDS, PANSS,side effects 65% At post-intervention, the acamprosate group did not differ significantly from the placebo group with respect to any of the outcomes (including side effects).No differences in side effects were observed between the two groups.A total of 16 adverse events were recorded, 7 in the placebo group (2 events reported by the same participant), 2 in the acamprosate group, and 7 events were deemed unrelated to study participation.
Nalmefene
Vasile et al., 2014 [50]*(N = 22) Single-arm, OL trialInpatients 45% 44 years (SD not reported) N = 22 (100%)(S: n = 22) None Not required Nalmefene 18 mg pro necessitate AP 24 weeks Week 24 None GGT Change in GGT CGI-S, GAF, IDTS-A, PANSS, side effects 82% A reduction in GGT levels, along with improved scores on the CGI-S, GAF, IDTS-A, and PANSS, were observed at post-treatment compared to baseline.Mild to moderate side effects (12 patients).

Abbreviations: AP: antipsychotics; ASI: addiction severity index; ASP: abstinence in study period; AUD: alcohol use disorder; AUDIT: alcohol use disorder identification test; AUS: alcohol use scale; BP: bipolar disorder; BSI: brief symptom inventory; CDA: consecutive days abstinent; CDT: carbohydrate-deficient transferrin; CDSS: Calgary Scale for Depression in Schizophrenia; CGI-S: clinical global impressions - severity; CUD: cocaine use disorder; DA: days abstinent; DB: double-blind; DD: drinking days; DH: days hospitalized; DDD: drinks per drinking day; DDI: days of drinking to intoxication; DDW: drinking days per week; DUS: drug use scale; DW: drinks per week; GAD: generalized anxiety disorder; GAF: global assessment of functioning; GGT: gamma-glutamyltransferase; GID: gender identity disorder; HDD: heavy drinking days; HSCL: Hopkins Symptom Checklist; IDTS-A: inventory of drug taking situations – alcohol focused version; MDD: major depressive disorder; OCDS: obsessive compulsive drinking scale; OL: open-label (unblinded); OPTNFS: outpatient psychiatric treatment not further specified; PANSS: positive and negative syndrome scale; PI: psychological intervention; PTSD: post traumatic stress disorder; QoH: quality of alcohol high; RCR: retrospective chart review; RCT: randomized controlled trial; RD: reduced drinking; S: schizophrenia; SAD: schizoaffective disorder; SGOT, serum glutamic-oxaloacetic transaminase; SGPT: serum glutamic pyruvic transaminase; SPD: schizoid personality disorder; TA: total abstinence ; TCQ: Tiffany Craving questionnaire; TDSP: total drinks in study period; TL: transaminase level; TLFB: Timeline Followback; UP: unspecified psychosis; UTS: urine toxicology screen; VAS: visual analog scale.

*conference abstract.