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. 2024 Mar 15;9(2):359–368. doi: 10.1016/j.synbio.2024.03.006

Table 1.

Inhibition constants of acarbose, acarstatin A and acarstatin B towards human salivary α-amylase and porcine pancreatic α-amylase.

Inhibitors Human salivary α-amylase
Porcine pancreatic α-amylase
Ki Inhibitory potency Ki Inhibitory potency
Acarbose 4.01 μM 6.54 μM
Acarstatin A 2.53 nM 1584 4.16 nM 1573
Acarstatin B 2.72 nM 1478 8.81 nM 742