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. 2024 Mar 20;14:1347402. doi: 10.3389/fonc.2024.1347402

Table 3.

RBPs and their role in inflammation and hematological malignancies.

RBP Function Role in Inflammation Role in Hematological Malignancies Clinical Implications Drugs/Inhibitors References
ZFP36 (TTP) mRNA destabilization Inhibits cytokine production
(TNF-α, IL-6)
Implicated in inflammation-induced cancer development and progression Potential tumor suppressor; Restoration may impair lymphoma development None specified (271, 272)
HuR (ELAVL1) mRNA stabilization Increases stability of pro-inflammatory cytokine mRNAs Associated with various cancers (e.g., breast, lung, ovarian) Cytoplasmic expression correlates with tumor size and grade; Potential therapeutic target HuR inhibitors (e.g., MS-444, H1N, Mitoxantrone, CMLD-2, Quercetin, dihydrotanshinone-I) (223, 273)
IGF2BPs (13) Regulate mRNA stability, translation, decay Stabilize pro-inflammatory genes in JAK/STAT, ErbB pathways Implicated in multiple cancers (e.g., B-ALL, breast, colon) Overexpression linked to tumor-associated inflammation; Potential therapeutic targets BTYNB,
C20H18BrN5OS,
Compound 7773, JX5, CWI 1-2
(274, 275)
RBM39 (CAPER) Pre-mRNA splicing; NFκB activation Regulates steroid hormone receptor-mediated transcription Associated with multiple malignancies (e.g., TNBC, AML) Higher expression in various cancers; Implication in NFκB activation E7820 (127, 276, 277)