Table 3.
MIC of compounds 3a-d and 4a-p against gram-negative and gram-positive bacteria.
Extract ID |
Gram positive |
Gram negative |
||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
Comd No. | MRSA | MIC μg/mL | En |
MIC μg/mL |
Sa | MIC μg/mL | K |
MIC μg/mL |
Se | MIC μg/mL | E. coli | MIC μg/mL |
3a | ++ | 256 | ++ | 32 | N | N | ++ | 128 | ++ | 64 | ++ | 128 |
3b | ++ | 256 | +++ | 16 | ++ | 64 | ++ | 128 | ++ | 64 | ++ | 128 |
3c | ++ | 256 | ++ | 64 | ++ | 64 | ++ | 128 | ++ | 128 | N | N |
3d | ++ | 256 | ++ | 32 | ++ | 64 | ++ | 128 | ++ | 128 | N | N |
4a | ++ | 256 | N | N | ++ | 32 | ++ | 128 | ++ | 128 | ++ | 128 |
4b | ++ | 256 | ++ | 32 | ++ | 32 | ++ | 128 | ++ | 128 | N | N |
4c | ++ | 128 | ++ | 32 | ++ | 32 | ++ | 128 | ++ | 128 | N | N |
4d | ++ | 128 | ++ | 32 | N | N | ++ | 128 | ++ | 128 | ++ | 128 |
4e | N | N | ++ | 32 | ++ | 64 | ++ | 128 | ++ | 128 | N | 128 |
4f | N | N | +++ | 16 | ++ | 64 | ++ | 128 | ++ | 128 | N | N |
4g | ++ | 128 | N | N | ++ | 64 | N | N | ++ | 128 | ++ | 128 |
4h | ++ | 128 | +++ | 16 | ++ | 64 | ++ | 128 | ++ | 128 | ++ | 128 |
4i | ++ | 128 | N | N | ++ | 64 | +++ | 16 | ++ | 128 | ++ | 128 |
4j | ++ | 128 | +++ | 16 | ++ | 64 | ++ | 128 | ++ | 128 | N | N |
4k | ++ | 128 | N | N | ++ | 64 | +++ | 16 | ++ | 128 | ++++ | 8 |
4l | ++ | 128 | ++ | 32 | ++ | 64 | N | N | ++ | 128 | ++ | 128 |
4m | ++ | 128 | ++ | 32 | ++ | 64 | +++ | 16 | ++ | 128 | ++ | 128 |
4n | ++ | 128 | ++ | 32 | +++ | 16 | +++ | 16 | ++ | 128 | ++++ | 8 |
4o | ++ | 128 | +++ | 16 | ++ | 64 | ++ | 128 | ++ | 128 | +++ | 16 |
4p | ++ | 128 | ++ | 32 | ++ | 64 | ++ | 128 | ++ | 128 | ++ | 128 |
DMSO -ve control |
N | N | N | N | N | N | N | N | N | N | N | N |
Amoxicillin +ve control |
+++ | 16 | +++ | 16 | +++ | 16 | +++ | 16 | +++ | 16 | +++ | 32 |
Se=Salmonella enteritidis; Sa = Staphylococcus aureus; MRSA = Methicillin-resistant Staphylococcus aureus. Ec = Escherichia coli, Pm=Proteus mirabilis, En = Enterococcus faecalis, K=Klebsiella pneumonia; N, not detected, DMSO is a negative control, Amoxicillin is a positive control Key to interpretation: >16 mm (+++++): very active. 10–15 mm (+++): active; less active; 6–10 mm (++): moderately active; 1–5 mm (+): inactive; (N): No inhibition zone.