Table 1.
TRP channel | Alternative name | Organism | Tissue distribution | TRP subfamily | Thermal sensitivitya | Activity range | Entropy change (ΔS) cal/mol∗K | Activation enthalpy (ΔH) kcal/mol | Q10b | Reference |
---|---|---|---|---|---|---|---|---|---|---|
TRPV1 | Vr1 | Rattus norvegicus (rat), Homo sapiens (human) | nociceptor neurons | Vanilloid | ≥42°C (40–45), T(0.5) = 51°C | 40.9°C-55.8 °Cc | 260 (at 30mV) | 90–100 | 16.8, 20 | Caterina et al.13, Yao et al.52, Tominaga, et al.54, Liu et al.55, Cheng et al.65 |
TRPV1(l) | TRPV1- long | Desmodus rotundus (vampire bat) | Dorsal root ganglion (DRG) and trigeminal ganglion (TG) neurons | Vanilloid | 40°C | ND | ND | ND | 12 | Gracheva et al.14 |
TRPV1(s) | TRPV1- short | Desmodus rotundus (vampire bat) | TG neurons | Vanilloid | 30°C | ND | ND | ND | 5 | Gracheva et al.14 |
TRPV2 | Vrl2 | Rattus norvegicus (rat), Homo sapiens (human) | nociceptor neurons, brain, spinal cord | Vanilloid | ≥52°C (50°C–53°C) | ND | 586 | 200 | 20.6 | Caterina et al.15 |
hTrpv3 | Vrl3 | Homo sapiens (human) | skin keratinocytes | Vanilloid | ≥33°C (34°C–38°C) | 33°C–50°C (Max 41°C–47°C) | ND | ND | 6.62 | Peier et al.123, Smith et al.124, Xu et al.125 |
hTrpv4 | OTRPC4, VR-OAC, Trp12, Vrl2 | Homo sapiens (human) | skin and dorsal root ganglion neurons, kidney, brain, liver, heart, hypothalamus | Vanilloid | ∼27°C–34°C | ND | ND | ND | 9.9 ± 3.8 | GÜler et al.73, Watanabe et al.126 |
TRPM8 | CMR1 | Homo sapiens (human) | DRG neurons, various organs | Melastatin | ≤23°C–25°C | 0°C-25°C | −384 | −112 | 24 | Brauchi et al.70, McKemy et al.127 |
TRPM3 | Mus musculus (mouse) | DRG and TG sensory neurons | Melastatin | ≥43°C | ND | ND | ND | 7.2 | Vriens et al.16 | |
TRPC5 | Mus musculus (mouse), Homo sapiens (human) | DRG neurons | Canonical | <37°C to >25°C | ND | ND | −40 | ND | Zimmermann et al.128 | |
Anktm1 | TRPA1 | Mus musculus (mouse), Homo sapiens (human) | DRG neurons | Ankyrin | ≤17°C | 0°C–17°C | −140 | −40 | 6 | Story et al.129 |
Chicken TRPA1 | TRPA1 | Gallus gallus domesticus (chicken) | DRG neurons | Ankyrin | 39.4°C | ND | ND | ND | ND | Saito et al.130 |
xtTRPA1 | TRPA1 | Xenopus tropicalis (Western clawed frog) | DRG neurons | Ankyrin | 39.7°C | ND | ND | ND | 59.24 ± 18 | Ohkita et al.131 |
xlTRPA1 | TRPA1 | Xenopus laevis (African clawed frog) | DRG neurons | Ankyrin | 36.2 ± 0.4°C | ND | ND | ND | ND | Saito et al.132 |
snTRPA1 | TRPA1 | Crotalus atrox (rattlesnake) | TG neurons | Ankyrin | 27.6°C | ND | ND | ND | 13.7 | Gracheva et al.133 |
python TRPA1 | TRPA1 | Python regius (python) | TG neurons | Ankyrin | 32.7°C | ND | ND | ND | ND | Gracheva et al.133 |
boa TRPA1 | TRPA1 | Corallus hortulanus (boa) | TG neurons | Ankyrin | 29.6°C | ND | ND | ND | ND | Gracheva et al.133 |
ratsnake TRPA1 | TRPA1 | Elaphe obsoleta lindheimeri (rat snake) | TG neurons | Ankyrin | 37.2°C | ND | ND | ND | 8.8 | Gracheva et al.133 |
Anole TRPA1 | TRPA1 | Anolis carolinensis (green anole) | TG neurons | Ankyrin | 33.9°C | ND | ND | ND | 45.71 ± 6 | Saito et al.134 |
A. allogus TRPA1 | TRPA1 | Anolis allogus (spanish flag anole) | Dorsal skin | Ankyrin | 33.5 ± 0.7°C | ND | ND | ND | ND | Akashi et al.135 |
A. homolechis TRPA1 | TRPA1 | Anolis homolechis (Habana anole) | Dorsal skin | Ankyrin | 36.4 ± 0.8°C | ND | ND | ND | ND | Akashi et al.135 |
A. sagrei TRPA1 | TRPA1 | Anolis sagrei (brown anole) | Dorsal skin | Ankyrin | 33.5 ± 0.7°C | ND | ND | ND | ND | Akashi et al.135 |
axTRPA1 | TRPA1 | Ambystoma mexicanum (axolotl) | Brain, lung, heart, stomach | Ankyrin | 39.7 ± 1.0°C | ND | ND | ND | ND | Oda et al.136 |
zTRPA1b | TRPA1 | Danio rerio (zebrafish) | Sensory neurons innervating skin and cranial sensory ganglia | Ankyrin | variable <10°C (cold); >25°C (heat) | ND | ND | ND | 8.2 ± 0.6 | Oda et al.137 |
olTRPA1 | TRPA1 | Oryzias latipes (medaka) | Ankyrin | variable | ND | ND | ND | ND | Oda et al.138 | |
trTRPA1 | TRPA1 | Takifugu rubripes (pufferfish) | Ankyrin | variable <8°C (cold); >25°C (heat) | ND | ND | ND | ND | Oda et al.139 | |
hTrpv4 | OTRPC4, VR-OAC, Trp12, Vrl2 | Homo sapiens (human) | skin and dorsal root ganglion neurons | Vanilloid | ∼27°C–34°C | ND | ND | ND | 9.9 ± 3.8 | GÜler et al.73, Watanabe et al.126 |
ceTRPA | Caenorhabditis elegans (nematode) | neurons, muscle, intestine, and epithelial cells | ≤17°C | ND | ND | ND | ND | Laursen et al.83 | ||
Painless | dAnktm1 | Drosophila melanogaster (fruit fly) | Peripheral neurons larval epidermis | Ankyrin | ∼39°C–42°C | ND | ND | ND | ND | Tracey et al.17 Sokabe et al.96 |
Pyrexia | Pyx-PA and Pyx-PB | Drosophila melanogaster (fruit fly) | embryos: peripheral nerves, central nerves, multidendritic neurons in larval epidermis; adults: sensory neurons around bristle eyes, bristle neurons along thorax, neurons in maxillary palps, proboscis, antennae | Ankyrin | ≥40°C | ND | ND | ND | Pyx-PA 18.145; Pyx-PB 15.329 | Lee et al.18, Neely et al.63 |
dTRPA1(A) | TrpA1-RI (Prom B, ex10a), dTrpA1, dANKTM1, DmTRPA1 | Drosophila melanogaster (fruit fly) | larval sensory neurons, adult proboscis | Ankyrin | 27°C-29°C | ND | ND | ND | 9 | Kang et al.19, Hamada et al.21, Rosenzweig et al.64, Viswanath et al.140 |
dTRPA1(D) | TrpA1-RG (Prom A, ex10a), dTrpA1, dANKTM1, DmTRPA1 | Drosophila melanogaster (fruit fly) | larval nociceptors | Ankyrin | ≥46°C, T(0.1) = 43°Cc, T(0.5) = 53.5 °Cc | 43-60 °Cc | 211c | 69c | 23,58c | Zhong et al.22 |
AgTRPA1 | Anopheles gambiae (African malaria mosquito) | antennae, head | Ankyrin | 25.2°C | ND | ND | ND | ND | Wang et al.25 | |
AsTRPA1(A) | Anopheles stephensi (Asian malaria mosquito) | antennae, head | Ankyrin | 30.3 ± 0.9°C | ND | ND | ND | 14,5 | Li et al.141 | |
AaTRPA1(B) | Aedes aegypti (yellow fever mosquito) | antennae, head | Ankyrin | 32 ± 0.8°C | ND | ND | ND | 20,7 | Li et al.141 | |
CpTRPA1(A) | Culex pipiens pallens (northern house mosquito) | antennae, head | Ankyrin | 21.8 ± 0.7°C | ND | ND | ND | 61,2 | Li et al.141 | |
BmTRPA1 | Bombyx mori (silk moth) | epidermlal non-neural cells of various tissues | Ankyrin | 21.6°C | 21.6°C–43.5°C | ND | ND | 20,5 | Saito et al.130 | |
HsTRPA | Am-HsTRPA | Apis mellifera (honeybee) | brain, leg, proboscis, antennae | Ankyrin | 33.9 ± 0.6°C | ND | ND | ND | 17.2 ± 4.0 | Kohno et al.28 |
RpTRPA5Bc | Rhodnius prolixus (kissing bug) | head, rostrum, legs, antennae, thorax, abdomen | Ankyrin | T(0.1) = 53°C; T(0.5) = 58.6°C | 50°C-68°C | 216 | 72 | 25 | c |
activation threshold temperature as determined in heterologous expression systems.
Q10 is the fold current increase over 10°C increase as a measure of sensitivity; the higher Q10 value, the more sensitivity to heat exhibited by the TRP channel.
experimental values determined in this study.