Table 2.
List Of GPCRS tested for agonist and antagonist activity
| GPCR | GPCR | GPCR |
| 5-HT1A | CysLT1 | Motilin |
| 5HT1B | CysLT2 | MrgD |
| 5-HT2A | D1 | MRGX1 |
| 5-HT2B | D2 | MRGX2 |
| 5-HT2C | D4 | NK1 |
| 5-HT4B | D5 | NK2 |
| 5-HT6 | DP | NK3 |
| A1 | EP1 | NMU1 |
| A2A | EP2 | NMU2 |
| A2B | EP3 | NOP |
| A3 | EP4 | NPBW1 |
| α1A | ETA | NTR1 |
| ADRA1A | ETB | OPRD1 |
| ADRA1B | FP | OPRK1 |
| ADRA1D (ñ2-79) | FPR1 | OPRM1 |
| ADRA2A | FPR2 | OT |
| ADRB1 | GABAB1b | OX1 |
| ADRB2 | GAL1 | OX2 |
| ADRB3 | GAL2 | P2Y1 |
| APJ | GCGR | P2Y11 |
| AT1 | Ghrelin | P2Y12 |
| BB1 | GIP | P2Y2 |
| BB2 | GLP-1 | P2Y4 |
| BB3 | GLP-2 | PAC1 |
| BDKR2 | GnRH | PAF |
| BLT1 | GPR103 | PK1 |
| C3aR | GPR109A | PK2 |
| C5aR | GPR14 | PRP |
| CaS | GPR39 | PTH1 |
| CB1 | GPR41 | PTH2 |
| CB2 | GPR43 | S1P1 |
| CCK1 | GPR54 | S1P2 |
| CCK2 | GPR68 | S1P3 |
| CCR1 | GPR91 | S1P4 |
| CCR10 | GPR99 | S1P5 |
| CCR2B | H1 | Secretin |
| CCR3 | H2 | sst2 |
| CCR4 | H3 | sst3 |
| CCR5 | IP1 | sst4 |
| CCR6 | LPA1 | sst5 |
| CCR7 | LPA3 | Thrombin-Activated PARs |
| CCR8 | LPA5 | TP |
| CCR9 | M1 | TRH |
| CGRP1 | M2 | Trypsin-Activated PARs |
| ChemR23 | M3 | TSH |
| CRF1 | M4 | V1A |
| CRF2 | M5 | V1B |
| CX3CR1 | MC2 | V2 |
| CXCR1 | MC4 | VPAC1 |
| CXCR2 | MC5 | VPAC2 |
| CXCR3 | MCHR1 | XCR1 |
| CXCR4 | MCHR2 | Y2 |
| CXCR5 | mGlu2 | Y4 |
| CXCR6 | mGlu1 |