| AbTACs | Antibody-based PROTACs |
| AURKs | Aurora kinases |
| AUTOTAC | Autophagy-targeting chimera |
| BBB | Blood–brain barrier |
| BTK | Bruton tyrosine kinase |
| c-MET | Cellular mesenchymal-to-epithelial transition factor |
| CNS | Central nervous system |
| CRBN | Cereblon |
| CLL | Chronic lymphocytic leukemia |
| CSF-1R | Colony-stimulating factor 1 receptor |
| CR | Complete response |
| dTAGs | Degradation tags |
| DC | Dendritic cell |
| DOR | Duration of response |
| EFS | Event-free survival |
| EGFR | Epidermal growth factor receptor |
| eTPD | Extracellular targeted protein degradation |
| FGFRs | Fibroblast growth factor receptors |
| HyT-PD | Hydrophobic tagging-based protein degradation |
| ICIs | Immune checkpoint inhibitors |
| IGF-1R | Insulin-like growth factor 1 receptor |
| IND | Investigational New Drug |
| LYTACs | Lysosome-targeting chimeras |
| LTR | Lysosome-targeting receptor |
| mAbs | Monoclonal antibodies |
| NMPA | National Medical Products Administration |
| NEK7 | NIMA-related kinase 7 |
| ORR | Overall response rate |
| AKT | Protein kinase B |
| POI | Protein of interest |
| PKIIs | Protein–kinase interaction inhibitors |
| PPI | Protein–protein interaction |
| PPIs | Protein–protein interactions |
| PROTACs | Proteolysis-targeting chimeras |
| RET | Proto-oncogene tyrosine protein kinase receptor |
| ROR1 | Receptor tyrosine kinase-like orphan receptor 1 |
| RTKs | Receptor tyrosine kinases |
| ROS1 | ROS proto-oncogene 1 |
| SMKIs | Small-molecule kinase inhibitors |
| TPD | Targeted protein degradation |
| TRK | Tropomyosin receptor kinase |
| TME | Tumor microenvironment |
| TAMs | Tumor-associated macrophages |
| FDA | U.S. Food and Drug Administration |
| UC | Urothelial carcinoma |