TABLE 8.

Nuclear receptor activation.

Fold activation	PXR	AhR	CAR3
100 μM ELP‐004	2.28	26.00	1.00
32 μM ELP‐004	1.60	11.18	0.06
10 μM ELP‐004	0.86	4.94	0.69
3.2 μM ELP‐004	1.18	1.86	0.66
1.0 μM ELP‐004	0.48	1.41	0.82
0.32 μM ELP‐004	1.21	1.09	0.48
EC50 (μM)	38.06	38.07	‐