| ADC | Antibody–drug conjugate |
| Ala | Alanine |
| BV | Brentuximab vedotin |
| Cit | Citrulline |
| Cys | Cysteine |
| DAR | Drug–Antibody Ratio |
| Dato-DXd | Datopotamab deruxtecan |
| DM1 | Mertansine/emtansine (maytansinoid) |
| DM4 | Soravtansine/ravtansine (maytansinoid) |
| DOX | Doxorubicin |
| DS-8201a | Trastuzumab deruxtecan |
| DXd | Exatecan derivative |
| EMA | European Medicines Agency |
| Fabs | Antigen-binding fragments |
| Fc | Fragment crystallizable region |
| FDA | Food and Drug Administration |
| G2 | Second growth phase |
| GO | Gemtuzumab ozogamicin |
| HER2 | Human epidermal growth factor receptor 2 |
| huC242-SPDB-DM4 | Cantuzumab ravtansine |
| Le(Y) | Anti-Lewis Y |
| Lys | Lysine |
| M | Mitosis |
| mAb | Monoclonal antibody |
| MC | Maleimidocaproyl |
| MK-2870 | Sacituzumab tirumotecan |
| MMAE | Monomethyl auristatin E |
| MRG002 | Human Epidermal Growth Factor Receptor 2 Positive Breast Cancer |
| MRG003 | Anti-Epidermal Growth Factor Receptor Antibody Drug Conjugate |
| NSCLC | Non-small cell lung cancer |
| PABC | P-aminobenzyloxycarbonyl |
| PBD | Pyrrolobenzodiazepine dimer |
| PEG | Polyethylene glycol |
| Phe | Phenylalanine |
| PK | Pharmacokinetics |
| RC48 | Disitamab vedotin |
| R-DXd | Raludotatug deruxtecan |
| SG | Sacituzumab govitecan |
| SN-38 | Active metabolite of iridotecan |
| SSC | Site-specific conjugation |
| T-DM1 | Trastuzumab emtansine conjugate DM1 |
| TNBC | Triple-negative breast cancer |
| Val | Valine |