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. 2024 Jun 26;25(13):6969. doi: 10.3390/ijms25136969
ADC Antibody–drug conjugate
Ala Alanine
BV Brentuximab vedotin
Cit Citrulline
Cys Cysteine
DAR Drug–Antibody Ratio
Dato-DXd Datopotamab deruxtecan
DM1 Mertansine/emtansine (maytansinoid)
DM4 Soravtansine/ravtansine (maytansinoid)
DOX Doxorubicin
DS-8201a Trastuzumab deruxtecan
DXd Exatecan derivative
EMA European Medicines Agency
Fabs Antigen-binding fragments
Fc Fragment crystallizable region
FDA Food and Drug Administration
G2 Second growth phase
GO Gemtuzumab ozogamicin
HER2 Human epidermal growth factor receptor 2
huC242-SPDB-DM4 Cantuzumab ravtansine
Le(Y) Anti-Lewis Y
Lys Lysine
M Mitosis
mAb Monoclonal antibody
MC Maleimidocaproyl
MK-2870 Sacituzumab tirumotecan
MMAE Monomethyl auristatin E
MRG002 Human Epidermal Growth Factor Receptor 2 Positive Breast Cancer
MRG003 Anti-Epidermal Growth Factor Receptor Antibody Drug Conjugate
NSCLC Non-small cell lung cancer
PABC P-aminobenzyloxycarbonyl
PBD Pyrrolobenzodiazepine dimer
PEG Polyethylene glycol
Phe Phenylalanine
PK Pharmacokinetics
RC48 Disitamab vedotin
R-DXd Raludotatug deruxtecan
SG Sacituzumab govitecan
SN-38 Active metabolite of iridotecan
SSC Site-specific conjugation
T-DM1 Trastuzumab emtansine conjugate DM1
TNBC Triple-negative breast cancer
Val Valine