Table 10.
Reaction Scheme | R1 | R2 | Compound | Yield (%) |
---|---|---|---|---|
5-OMe | H | 59a | 74 | |
5-Me | H | 59b | 80 | |
5-F | H | 59c | 86 | |
5-Cl | H | 59d | 66 | |
5-Br | H | 59e | 73 | |
5-I | H | 59f | 77 | |
6-F | H | 59g | 90 | |
6-Cl | H | 59h | 90 | |
6-Br | H | 59i | 76 | |
4-Br | H | 59j | 59 | |
7-Me | H | 59k | 76 | |
H | 2-Me | 59l | 75 |