| Entry |
Substrates
(2a–p) |
Products
(3a–p) |
m.p. a
(°C) |
Yield b
% |
| 1 |
2a
|
3a
|
186–188 | 79 |
| 2 |
2b
|
3b
|
183–184 | 62 |
| 3 |
2c
|
3c
|
193–195 | 81 |
| 4 |
2d
|
3d
|
183–185 | 75 |
| 5 |
2e
|
3e
|
168–179 | 77 |
| 6 |
2f
|
3f
|
189–191 | 73 |
| 7 |
2g
|
3g
|
195–197 | 65 |
| 8 |
2h
|
3h
|
178–179 | 82 |
| 9 |
2i
|
3i
|
168–170 | 61 |
| 10 |
2j
|
3j
|
199–201 | 85 |
| 11 |
2k
|
3k
|
210–212 | 78 |
| 12 |
2l
|
3l
|
189–191 | 68 |
| 13 |
2m
|
3m
|
167–169 | 71 |
| 14 |
2n
|
3n
|
179–181 | 77 |
| 15 |
2o
|
3o
|
205–207 | 84 |
| 16 |
2p
|
3p
|
223–225 | 80 |
| a Melting point of products 3a–p; b isolated yield of products 3a–p. | ||||
2a
3a
2b
3b
2c
3c
2d
3d
2e
3e
2f
3f
2g
3g
2h
3h
2i
3i
2j
3j
2k
3k
2l
3l
2m
3m
2n
3n
2o
3o
2p
3p