Determination of MIC's of 6H-1,2-oxazin-6-onesa.
| 6H-1,2-oxazin-6-ones | 43 300 | SARM 3 | SARM 4 | SARM 5 | 25 922 | ||
|---|---|---|---|---|---|---|---|
| R1 | R2 | ||||||
| 1 | 4-Cl | 4-Me | 3.125 | — | 3.125 | 3.125 | — |
| 2 | 4-H | 4-Me | 200 | 200 | 200 | 200 | 200 |
| 3 | 4-Cl | 4-Cl | 100 | — | — | — | — |
| 4 | 4-Me | 4-Cl | 12.5 | 12.5 | 12.5 | 12.5 | 12.5 |
| 6 | 4-Me | 4-Me | 50 | 50 | — | 50 | — |
| 8 | 4-Me | 4-OMe | 25 | 25 | 25 | 25 | 25 |
| Gentamicin | 2 | 1 | 2 | 2 | 1 | ||
| Linezolid | 4 | 4 | 8 | 8 | — | ||
| Trimethoprim | 1 | 1 | 2 | 2 | — | ||
MRSA ATCC 43300, clinical Isolates MRSA 3, MRSA 4, MRSA5, E. coli ATCC 25922. (—): no activity.