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. 2024 Jul 26;4:1411935. doi: 10.3389/fbinf.2024.1411935

TABLE 3.

Potential drug targets in Escherichia coli that confer antibiotic resistance.

S/No Antimicrobial resistance mechanism Genes/proteins
1 Antibiotic activation enzyme KatG
2 Antibiotic resistance gene cluster, cassette, or operon MarA, MarB, MarR
3 Antibiotic target in susceptible species Alr, Ddl, dxr, EF-G, EF-Tu, folA, Dfr, folP, gyrA, gyrB, inhA, fabI, Iso-tRNA, MurA, rho, rpoB, rpoC, S10p, S12p
4 Antibiotic target protection protein BcrC
5 Efflux pump conferring antibiotic resistance AcrAB-TolC, AcrZ, EmrAB-TolC, MacA, MacB, MdfA/Cmr, MdtEF-TolC, MdtL, TolC/OpmH
6 Gene conferring resistance via absence gidB
7 Protein altering cell wall charge conferring antibiotic resistance PgsA
8 Regulator modulating expression of antibiotic resistance genes AcrAB-TolC, EmrAB-TolC, GadE, H-NS, OxyR