Table 2.
Entry | TAME | FABP5/3 SI | FABP5 KI (μM) | FABP5/7 SI |
---|---|---|---|---|
| ||||
1 | α-16 | 41.3 | 1.30 ± 0.28 | 16.7 |
2 | α-21 | 36.2 | 1.75 ± 0.07 | 0.47 |
3 | α-1 | 38.0 | 0.12 ± 0.02 | 4.5 |
4 | γ-12 | 32.3 | 0.79 ± 0.08 | 7.0 |
5 | α-12 | 26.9 | 0.87 ± 0.06 | 3.8 |
6 | α-5 | 16.7 | 0.36 ± 0.05 | 1.6 |
7* | L3 | 14.7 | 1.72 ± 0.12* | 8.3 |
8 | α-22 | 14.2 | 1.83 ± 0.27 | 4.2 |
9 | α-8 | 13.0 | 0.59 ± 0.08 | 0.56 |
10 | α-7 | 12.4 | 0.44 ± 0.05 | 4.5 |
11 | α-2 | 11.7 | 0.29 ± 0.01 | 0.41 |
12 | α-10 | 11.0 | 0.74 ± 0.06 | 0.95 |
13 | α-6 | 9.8 | 0.41 ± 0.15 | 2.2 |
14 | γ-9 | 9.0 | 0.89 ± 0.25 | 2.1 |
15 | γ-6 | 5.4 | 1.26 ± 0.12 | 1.4 |
16 | α-4 | 4.8 | 0.33 ± 0.06 | 2.9 |
17 | α-9 | 4.7 | 0.72 ± 0.08 | 1.4 |
18 | γ-102 | 4.2 | 1.39 ± 0.07 | 0.64 |
19 | α-15 | 3.7 | 1.30 ± 0.09 | 0.68 |
20 | γ-13 | 3.4 | 1.77 ± 0.02 | 2.0 |
Ki values represent an average ± S.E. of at least three independent experiments.
Ki values from Reference [34].