Table 3. Inhibition constants (Ki) for triclosan binding to wild-type and mutant PfENR.
Enzyme | Inhibition constant (Ki) (nM) |
---|---|
Wild-type | 0.03 (±0.001) |
A217V | 232.0 (±5.0) |
A217G | 0.57 (±0.05) |
N218A | 2.10 (±0.10) |
N218D | 1.50 (±0.04) |
M281A | 9.34 (±0.81) |
M281T | 10.0 (±0.89) |
F368A | 7.20 (±0.90) |
F368I | 6.30 (±0.56) |