Table 1.
Pharmacological drugs utilized for RVM microinjection experiments
| Pharmacologic | Target | Company | Catalog # | Concentration | Solution |
|---|---|---|---|---|---|
| ICI 182,780 | ER antagonist; GPER agonist | Tocris Bioscience | 1047 | 0.2–20 µM | 0.03% ethanol; 0.9% saline |
| Letrozole | Aromatase inhibitor | Selleckchem | S1235 | 350 µM–3.5 mM | 2% DMSO; 0.9% saline |
| MPP | ER-α antagonist | Tocris Bioscience | 1991 | 10–300 nM | 2% DMSO; 0.9% saline |
| PHTPP | ER-β antagonist | Tocris Bioscience | 2662 | 1 µM | 2% DMSO; 0.9% saline |