Table 3. The IC50 values and selectivities of DC01, DC24 and fasudil on ROCKs.
| Compd. | IC50 (μM) | Selectivity | |
|---|---|---|---|
| ROCK1 | ROCK2 | ||
| DC01 | 0.754 | 1.015 | — |
| DC24 | 6.354 | 0.124 | 51.24 |
| Fasudil | 0.358 | 0.158 | 2.27 |
| Compd. | IC50 (μM) | Selectivity | |
|---|---|---|---|
| ROCK1 | ROCK2 | ||
| DC01 | 0.754 | 1.015 | — |
| DC24 | 6.354 | 0.124 | 51.24 |
| Fasudil | 0.358 | 0.158 | 2.27 |