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. 2024 Aug 1;15(10):3576–3596. doi: 10.1039/d4md00438h

Table 3. The IC50 values and selectivities of DC01, DC24 and fasudil on ROCKs.

Compd. IC50 (μM) Selectivity
ROCK1 ROCK2
DC01 0.754 1.015
DC24 6.354 0.124 51.24
Fasudil 0.358 0.158 2.27