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. 2024 Mar 28;67(7):5421–5436. doi: 10.1021/acs.jmedchem.3c01993

Table 2. Aggregation Temperature (Tagg) for HUP-46, KYP-2091, and KYP-2112 in PREP and PREP Mutantsa.

Tagg (°C) hPREP Asn483Ala Leu499Cys Tyr471Ala
DMSO 48.9 ± 0.4 47.8 ± 0.4 47.7 ± 0.4 47.2 ± 0.5
HUP-46 53.2 ± 1.5 48.5 ± 0.4 48.3 ± 0.4 n.d.
KYP-2091 52.5 ± 1.0 49.3 ± 1.2 50.6 ± 4.6 47.8 ± 0.8
KYP-2112 52.2 ± 1.3 50.6 ± 1.0 54.2 ± 0.9 50.5 ± 0.5
a

n.d.: not detected.