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. 2024 Aug 7;40(4):533–540. doi: 10.1007/s43188-024-00259-8

Table 4.

Cellular Effects of DRD2 antagonists

Compound Cancer cells Effects Reference
Thioridazine Cancer stem cells from HCT116 Antitumor effect [47]
Thioridazine Cervical carcinoma SiHa Cell death [53]
Thioridazine Triple-negative breast cancer cells STAT3 inhibition [21]
Thioridazine Cervical cancer Akt, PI3K inhibition [54]
Thioridazine Leukemia cell mitochondrial Apoptotic pathway [55]
Haloperidol Glioblastoma ERK signaling↑ [58]
Domperidone Triple-negative breast Cancer cells ROS, JAK/STAT3 Signaling↑ [60]
Domperidone Small cell lung cancer cells Cell growth↑ [35]