Table 1.
Targets of Activity-Based Probes and Competition Experiments
| Protein ID | Annotation | Essential | Competed by 21 | Competed by 22 | Salinipostin A |
|---|---|---|---|---|---|
| PF3D7_1038900 | Esterase (PfMAGL) | Yes | Yes | No | Yes |
| PF3D7_0805000 | α/β hydrolase | No | No | No | Yes |
| PF3D7_0709700 | lysophospholipase (PfPARE) | No | Yes | Yes | Yes |
| PF3D7_1120400 | α/β hydrolase (abH12) | Yes | No | Yes | No |
| PF3D7_0619300 | unknown function | No | No | Yes | No |
| PF3D7_1116100 | serine esterase | No | No | No | Yes |
| NCEH 1 | Neutral cholesterol ester hydrolase 1 | N/A | Yes | Yes | N/A |
| AChE | Acetylcholinesterase | N/A | No | No | N/A |