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. 2001 Aug;75(16):7462–7469. doi: 10.1128/JVI.75.16.7462-7469.2001

TABLE 4.

Association of viral genotype with levels of reduced susceptibility to lopinavir

Mutation No. of occurrences Pa for cutoff of fold lopinavir IC50
4 10 20 40
L10F/I/R/V 45 0.0013 0.0013 0.0261 ns
K20M/R 13 ns ns 0.0028 ns
L24I 8 ns ns ns ns
M46I/L 27 ns ns ns ns
F53L 9 ns ns 0.0479 0.0173
I54L/T/V 27 <0.0001 <0.0001 <0.0001 0.0016
L63P 49 0.0371 0.0160 ns ns
A71I/L/V/T 35 0.0137 0.0301 ns ns
V82A/F/T 26 <0.0001 <0.0001 0.0005 0.0011
I84V 14 0.0121 ns ns ns
L90M 32 ns ns ns ns
a

P values <0.0075 were considered statistically significant; P values between 0.05 and 0.0075 were considered marginally significant; P values >0.05 were considered not significant (ns). 

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