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. 2024 Oct 11;13(10):2511–2523. doi: 10.21037/tlcr-24-273

Table 2. Drug dose modification.

Characteristics Subgroups N (%)
Dose reduction EGFR-TKI 0/44 (0.0)
MET-TKI 6/44 (13.6)
Drug discontinuation Both drugs 13/44 (29.5)
MET-TKI only 10/44 (22.7)
Cause of discontinuation of both drugs Pneumonitis 9/13 (69.2)
Hypersensitivity 2/13 (15.4)
Mediastinitis 1/13 (7.7)
Recurrent cellulitis 1/13 (7.7)
Cause of discontinuation of MET-TKI Hypersensitivity 5/10 (50.0)
Generalized pain 2/10 (20.0)
Hepatitis 2/10 (20.0)
Deep vein thrombosis 1/10 (10.0)
Discontinuation rate
per drug
EGFR-TKI
• 1st or 2nd generation 4/9 (44.4)
• 3rd generation 19/35 (54.3)
MET-TKI
• Savolitinib 19/31 (61.3)
• Crizotinib 3/11 (27.3)
• Capmatinib 1/2 (50.0)

TKI, tyrosine kinase inhibitor.