TABLE 2.
Pharmacological profile of α‐ and β‐agonists on inhibitory motor responses in the rat colon.
Agonists | Antagonists that block the inhibitory response | Antagonists that do not block the inhibitory response |
---|---|---|
Phenylephrine (α‐adrenoceptor agonist) |
Phentolamine: α‐adrenoceptor blocker Apamin: sKCa blocker Prazosin: α1‐adrenoceptor blocker RS17053: α1A‐adrenoceptor blocker a | Propranolol: β‐adrenoceptor blocker Yohimbine: α2‐adrenoceptor blocker |
Isoprenaline (β‐adrenoceptor agonist) |
Propranolol: β‐adrenoceptor blocker | Phentolamine: α‐adrenoceptor blocker |
Preferential α1A as it might also block α1D‐adrenoceptor.