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. 2024 Sep 30;37(1):e14921. doi: 10.1111/nmo.14921

TABLE 2.

Pharmacological profile of α‐ and β‐agonists on inhibitory motor responses in the rat colon.

Agonists Antagonists that block the inhibitory response Antagonists that do not block the inhibitory response

Phenylephrine

(α‐adrenoceptor agonist)

Phentolamine: α‐adrenoceptor blocker Apamin: sKCa blocker Prazosin: α1‐adrenoceptor blocker RS17053: α1A‐adrenoceptor blocker a Propranolol: β‐adrenoceptor blocker Yohimbine: α2‐adrenoceptor blocker

Isoprenaline

(β‐adrenoceptor agonist)

Propranolol: β‐adrenoceptor blocker Phentolamine: α‐adrenoceptor blocker
a

Preferential α1A as it might also block α1D‐adrenoceptor.