Table 3. Relative Binding Free Energies (RBFEs) (in Kcal Mol–1) for Ligand Pairs Studied Here.
system | ligands | RBFEcalc.a | RBFEexp. |
---|---|---|---|
thrombin | B5–B1a | –0.97 ± 0.4 | –0.6141 |
scytalone dehydratase | C3d-C5d | –1.59 ± 0.5 | –1.9839 |
factor Xa | IID-IIE | –2.46 ± 0.5 | –1.9842 |
BACE1 | C4j-C4b | 0.32 ± 0.6 | –0.6143 |
BTK | S8–S11 | –4.08 ± 0.7 | –1.9144 |
Uncertainties are calculated over three simulation repeats.