Table 4.
Agonists and antagonists of TRP channels.
| agonists | antagonists | Applications | Ref | |
|---|---|---|---|---|
| TRPA1 | Mustard oil, Cinnamaldehyde | HC-030031, A-967079 | Pain, inflammation | 79 |
| TRPV1 | Capsaicin, Heat, Resiniferatoxin | Capsazepine, Capsaicin (high dose) | Pain | 80 |
| TRPV4 | 4α-PDD, GSK1016790A | HC-067047, RN-1734 | Inflammation | 81 |
| TRPM8 | Menthol, Eucalyptol, Cubebol | AMG-333, Cannabidivarin, PF-05105679 | Pain | 15 |