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. 2022 Jul 1;149(7):2771–2782. doi: 10.1007/s00432-022-04149-0

Table 2.

List of compounds used in Phase II trials (randomized and single-arm trials), divided by main classes of drugs

Chemotherapy Targeted agents Immunotherapy Cellular therapy
Tyrosine kinase inhibitors (TKIs) Other

13‐Deoxy, 5‐iminodoxorubicin (GPX‐150)

Aldoxorubicin

Amrubicin

Bendamustin

Brostallicin

Dacarbazine

Docetaxel

Doxorubicin

Eribulin

Evofosfamide

Exatecan

Gemcatabine

Ifosfamide

Ixabepilone

Liposomal doxorubicin

Lurbinectedin

Non-pegylated liposomal doxorubicin

Paclitaxel

Pemetrexed

Plitidepsin

Soblidotin

Thalidomide

Trabectedin

Trofosfamide

Alisertib

Anlotynib

Axitinib

Brivanib

Cediranib

Crizotinib

Dasatinib

ENMD-2076

Gefitinib

Pazopanib

Regorafenib

Sorafenib

Sunitinib

Tivozanib

Aflibercept

Bevacizumab

Conatumumab

Ganetespib

Letrozole

Olaratumab

Ontuxizumab

Palbociclib

Panobinbostat

Perifosine

Ridaforolimus

Selumetinib

Sirolimus

Tazemetostant

Temsirolimus

Thrombospondin-1-Mimetic Angiogenesis Inhibitor ABT-510

Trebananib

Vorinostat

Nivolumab

Pembrolizumab

Talimogene laherparepvec (T-VEC)

NY-ESO-1c259T Cells