TABLE 4.
The inhibitory effect of BST-4 on other members of the BET and STAT families.
Targets | IC50 (μM) | Targets | IC50 (μM) |
---|---|---|---|
BRD2 | >10 | STAT4 | >10 |
BRD3 | >10 | STAT5a | >10 |
BRDT | >10 | STAT5b | >10 |
STAT1 | >10 | STAT6 | >10 |
STAT2 | >10 |
The inhibitory effect of BST-4 on other members of the BET and STAT families.
Targets | IC50 (μM) | Targets | IC50 (μM) |
---|---|---|---|
BRD2 | >10 | STAT4 | >10 |
BRD3 | >10 | STAT5a | >10 |
BRDT | >10 | STAT5b | >10 |
STAT1 | >10 | STAT6 | >10 |
STAT2 | >10 |