TABLE 4.
The inhibitory effect of BST-4 on other members of the BET and STAT families.
| Targets | IC50 (μM) | Targets | IC50 (μM) |
|---|---|---|---|
| BRD2 | >10 | STAT4 | >10 |
| BRD3 | >10 | STAT5a | >10 |
| BRDT | >10 | STAT5b | >10 |
| STAT1 | >10 | STAT6 | >10 |
| STAT2 | >10 |
The inhibitory effect of BST-4 on other members of the BET and STAT families.
| Targets | IC50 (μM) | Targets | IC50 (μM) |
|---|---|---|---|
| BRD2 | >10 | STAT4 | >10 |
| BRD3 | >10 | STAT5a | >10 |
| BRDT | >10 | STAT5b | >10 |
| STAT1 | >10 | STAT6 | >10 |
| STAT2 | >10 |