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. 2025 Apr 1;16:1556990. doi: 10.3389/fimmu.2025.1556990

Table 5.

Summarize the regulatory factors involved in Nrf2/HO-1 and HIF-1α-mediated pyroptosis in OA.

Regulatory element Signaling Pathway Biological function Animal models Reference
Oroxylin A Lcp1/HIF-1α Decreased subchondral bone remodeling and slowed cartilage degeneration Mice (130)
PD184352 Nrf2/HO-1 Anti-inflammatory and antioxidant effects Mice (171)
Myrislignan Nrf2/HO-1 Inhibits inflammation and oxidative stress Rats (172)
HMGB1 HO-1/VEGF Inhibits synovial angiogenesis Human FLS (176)
Silence HIF-1α HIF-1α/NLRP3 Inhibit pyroptosis of FLS Rats (177)
Agnuside(AGN) HIF-1α/NLRP3 Relieves synovitis and fibrosis in KOA Rats (178)