Table 2.
TEAE(≥ 20%) in the SS
| TEAEs, n (%) | 40 mg BID (n = 4) | 60 mg BID (n = 3) | 80 mg BID (n = 4) | Total (n = 11) | ||||
|---|---|---|---|---|---|---|---|---|
| Any grade | ≥ Grade 3 | Any grade | ≥ Grade 3 | Any grade | ≥ Grade 3 | Any grade | ≥ Grade 3 | |
| Any TEAEs | 4 (100) | 1 (25.0) | 3 (100) | 2 (66.7) | 4 (100) | 2 (50.0) | 11 (100) | 5 (45.5) |
| Hypertriglyceridemia | 1 (25.0) | 2 (66.7) | 1 (33.3) | 3 (75.0) | 2 (50.0) | 6 (54.5) | 3 (27.3) | |
| Neutropenia | 1 (25.0) | 1 (33.3) | 3 (75.0) | 5 (45.5) | ||||
| Hypoalbuminemia | 2 (50.0) | 2 (66.7) | 1 (25.0) | 5 (45.5) | ||||
| Hypoproteinemia | 1 (25.0) | 2 (66.7) | 2 (50.0) | 5 (45.5) | ||||
| Thrombocytopenia | 2 (50.0) | 1 (25.0) | 2 (66.7) | 1 (33.3) | 1 (25.0) | 5 (45.5) | 2 (18.2) | |
| Abnormal T-wave on electrocardiogram | 0 | 1 (33.3) | 3 (75.0) | 4 (36.4) | ||||
| Leukopenia | 0 | 1 (33.3) | 3 (75.0) | 4 (36.4) | ||||
| Diarrhea | 0 | 1 (33.3) | 3 (75.0) | 4 (36.4) | ||||
| Fatigue | 1 (25.0) | 1 (33.3) | 2 (50.0) | 4 (36.4) | ||||
| Anemia | 1 (25.0) | 1 (33.3) | 2 (50.0) | 4 (36.4) | ||||
| Elevated α-hydroxybutyrate dehydrogenase | 1 (25.0) | 1 (33.3) | 1 (25.0) | 3 (27.3) | ||||
| Elevated low-density lipoprotein | 1 (25.0) | 2 (66.7) | 0 | 3 (27.3) | ||||
| Urinary white blood cell positivity | 1 (25.0) | 1 (33.3) | 1 (25.0) | 3 (27.3) | ||||
| Abnormal ST segment on electrocardiogram | 0 | 1 (33.3) | 2 (50.0) | 3 (27.3) | ||||
| Nausea | 0 | 1 (33.3) | 2 (50.0) | 3 (27.3) | ||||
| Lymphopenia | 0 | 1 (33.3) | 2 (50.0) | 3 (27.3) | ||||
| Hyperuricemia | 1 (25.0) | 1 (33.3) | 1 (25.0) | 3 (27.3) | ||||
| Hypercholesterolemia | 1 (25.0) | 1 (33.3) | 1 (25.0) | 3 (27.3) | ||||
| Hyperglycemia | 1 (25.0) | 0 | 2 (50.0) | 1 (25.0) | 3 (27.3) | 1 (9.1) | ||