| 6-CF | 6-Carboxyfluorescein |
| ABC | ATP-binding cassette |
| ACE | Angiotensin-converting enzyme |
| ARBs | Angiotensin II receptor blockers |
| BBB | Blood–brain barrier |
| BCRP | Breast cancer resistant protein |
| BMECs | Human brain microvascular endothelial cells |
| CHO | Chinese hamster ovary cells |
| ciPTEC | Conditionally immortalized proximal tubule epithelial cells |
| CKD | Chronic kidney disease |
| CKD-MBD | Chronic kidney disease—mineral and bone disorder |
| CKD-REIN | Chronic Kidney Disease—Renal Epidemiology and Information Network |
| CNS | Central nervous system |
| CYP2E1 | Cytochrome P450 2E1 |
| DOACs | Direct oral anticoagulants |
| EPO | Erythropoietin |
| ES | Estrone sulfate |
| GERD | Gastroesophageal reflux disease |
| HEK293 | Human embryonic kidney cells |
| HK-2 | Human kidney-2 cells |
| HMG-CoA | 3-Hydroxy-3-methylglutaryl-coenzyme A |
| hOAT | Human organic anion transporter |
| HSA | Human serum albumin |
| HUVEC | Human umbilical vein endothelial cells |
| IS | Indoxyl sulfate |
| LLC-PK1 | Porcine kidney 1 epithelial cells |
| MDCK | Madin–Darby canine kidney cells |
| MRP | Multidrug resistance protein |
| MTX | Methotrexate |
| NSAIDs | Non-steroidal anti-inflammatory drugs |
| OAT | Organic anion transporter |
| OATP | Organic anion transporting polypeptide |
| PAH | p-Amminohippuric acid |
| PBUTs | Protein-bound uremic toxins |
| PCS | p-Cresyl sulfate |
| PEPT1 | Peptide transporter 1 |
| P-gp | P-Glycoprotein |
| PPIs | Proton pump inhibitors |
| rOAT | Rat organic anion transporter |
| S2-cells | Immortalized cell line derived from the second segment of mice proximal tubule |
| SLC | Solute carrier transporter |
| SULT1A1 | Sulfotransferase 1A1 |
| TAT | Tyrosine aminotransferase |
| UT | Uremic toxin |
| VKA | Vitamin K antagonist |